Compile Data Set for Download or QSAR
Found 27 of ic50 data for polymerid = 50004933
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))TBA
LigandPNGBDBM643202(US20240002380, Example 70)copy SMILES
Affinity DataIC50: 250nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))TBA
LigandPNGBDBM643187(US20240002380, Example 24)copy SMILES
Affinity DataIC50: 250nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))TBA
LigandPNGBDBM643186(US20240002380, Example 22)copy SMILES
Affinity DataIC50: 250nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))TBA
LigandPNGBDBM643193(US20240002380, Example 48)copy SMILES
Affinity DataIC50: 250nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))TBA
LigandPNGBDBM643189(US20240002380, Example 36)copy SMILES
Affinity DataIC50: 250nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))TBA
LigandPNGBDBM643200(US20240002380, Example 62)copy SMILES
Affinity DataIC50: 250nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))TBA
LigandPNGBDBM643179(US20240002380, Example 5)copy SMILES
Affinity DataIC50: 250nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))TBA
LigandPNGBDBM643180(US20240002380, Example 6)copy SMILES
Affinity DataIC50: 250nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))TBA
LigandPNGBDBM643181(US20240002380, Example 10)copy SMILES
Affinity DataIC50: 250nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))TBA
LigandPNGBDBM643199(US20240002380, Example 59)copy SMILES
Affinity DataIC50: 250nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))TBA
LigandPNGBDBM643196(US20240002380, Example 54)copy SMILES
Affinity DataIC50: 250nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))TBA
LigandPNGBDBM643184(US20240002380, Example 17)copy SMILES
Affinity DataIC50: 250nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))TBA
LigandPNGBDBM50366239(CHEMBL1961797)copy SMILEScopy InChI
Affinity DataIC50: 620nMAssay Description:REV-ERB-alpha mediated transcriptional suppression at Bmal1 promoter in HEK293 cell reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445N00PubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))TBA
LigandPNGBDBM50366238(CHEMBL1961796)copy SMILEScopy InChI
Affinity DataIC50: 670nMAssay Description:Agonist activity at Rev-Erbalpha expressed in HEK293 cells coexpressing Gal4 ligand binding domain assessed as inhibition of transcription after 24 h...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D21ZPZPubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))TBA
LigandPNGBDBM50366238(CHEMBL1961796)copy SMILEScopy InChI
Affinity DataIC50: 670nMAssay Description:Increased REV-ERB-alpha LBD dependent repressor activity in HEK293 cell reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445N00PubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))TBA
LigandPNGBDBM50366238(CHEMBL1961796)copy SMILEScopy InChI
Affinity DataIC50: 710nMAssay Description:REV-ERB-alpha mediated transcriptional suppression at Bmal1 promoter in HEK293 cell reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445N00PubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))TBA
LigandPNGBDBM50366239(CHEMBL1961797)copy SMILEScopy InChI
Affinity DataIC50: 790nMAssay Description:Increased REV-ERB-alpha LBD dependent repressor activity in HEK293 cell reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445N00PubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))TBA
LigandPNGBDBM643201(US20240002380, Example 68)copy SMILES
Affinity DataIC50: 1.00E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))TBA
LigandPNGBDBM643177(US20240002380, Example 3)copy SMILES
Affinity DataIC50: 1.00E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))TBA
LigandPNGBDBM643183(US20240002380, Example 14)copy SMILES
Affinity DataIC50: 1.00E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))TBA
LigandPNGBDBM643194(US20240002380, Example 49)copy SMILES
Affinity DataIC50: 1.00E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))TBA
LigandPNGBDBM643192(US20240002380, Example 46)copy SMILES
Affinity DataIC50: 1.00E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))TBA
LigandPNGBDBM643182(US20240002380, Example 13)copy SMILES
Affinity DataIC50: 1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))TBA
LigandPNGBDBM643198(US20240002380, Example 57)copy SMILES
Affinity DataIC50: 1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))TBA
LigandPNGBDBM643191(US20240002380, Example 45)copy SMILES
Affinity DataIC50: 1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))TBA
LigandPNGBDBM643185(US20240002380, Example 21)copy SMILES
Affinity DataIC50: 1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))TBA
LigandPNGBDBM643197(US20240002380, Example 56)copy SMILES
Affinity DataIC50: 1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails